APP-FUBINACA

APP-FUBINACA

APP-FUBINACA
Systematic (IUPAC) name
N-(1-amino-3-phenyl-1-oxopropan-2-yl)-1-[(4-fluorophenyl)methyl]-1H-indazole-3-carboxamide
Identifiers
CAS Registry Number
PubChem CID:
Chemical data
Formula C24H21FN4O2
Molecular mass 416.5 g/mol

APP-FUBINACA is an indazole-based synthetic cannabinoid that has been sold online as a designer drug.[1] Pharmacological testing showed APP-FUBINACA to have only moderate affinity for the CB1 receptor, with a Ki of 708 nM, while its EC50 was not tested.[2]

Legality

Sweden's public health agency suggested to classify APP-FUBINACA as hazardous substance on March 24, 2015.[3]

See also

References

  1. ^ "APP-FUBINACA". Cayman Chemical. Retrieved 15 July 2015. 
  2. ^ Buchler IP et al, INDAZOLE DERIVATIVES. WO 2009/106982
  3. ^ "Fler ämnen föreslås bli klassade som narkotika eller hälsofarlig vara". Folkhälsomyndigheten. Retrieved 16 July 2015.